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一、药化、抗菌素组本组共报告论文37篇,其中综述报告5篇;有15个省、市的代表参加报告。综述报告对当前国际上受人注意的一些理论问题作了介绍,如药物的定量构效关系,药物的构型,构象与生物活性的关系,体内金属离子与药物生物活性间的关系以及量子力学在药物化学中的应用等等,引起了到会同志们的兴趣。这些问题的探讨将为今后的新药设计提供依据。从各位代表所作的报告中可以看出,对近年来在国际上受人重视的一些课题如抗癌药,抗疟药、抗血吸虫药以及前列腺素类似物等等,在我国都已开展了
First, medicine, antibiotic group This group reported a total of 37 papers, including 5 review reports; 15 provinces, municipalities to participate in the report. The review report introduces some current international attention issues such as the quantitative structure-activity relationship of drugs, the conformation of drugs, the relationship between conformation and biological activity, the relationship between the metal ions in the body and the bioactivity of drugs, and the quantum mechanics The application in medicinal chemistry and so on, has aroused the interest of comrades in the meeting. The discussion of these issues will provide the basis for the future design of new drugs. As can be seen from the reports made by the deputies, some topics that have drawn international attention in recent years such as anti-cancer drugs, anti-malaria drugs, anti-schistosome drugs and prostaglandin analogues have all been carried out in our country