Caged Circular Antisense Oligonucleotides for Photomodulation of RNA Digestion and Gene Expression

来源 :第九届IUPAC化学生物学国际研讨会暨第八届世界华人药物化学研讨会 | 被引量 : 0次 | 上传用户:liyang0ly
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  In the thesis,we synthesized three 20mer caged circular asODNs(R20,R20B2 and R20B4) with a photocleavable linker and an amide bond linker between two 10mer ODNs.With these caged circular asODNs,RNA binding affinity and its digestion by RNase H were readily photomodulated.RNA cleavage rates were upregulated about 43-,25-and 15-fold for R20,R20B2 and R20B4,respectively,upon light-activation in vitro.
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