Antagonists相关论文
Dechloranes are a group of halogenated flame retardants with a basic bicyclo[2.2.1]heptene,including Dechlorane Plus (DP......
Integrins are transmembrane receptors that have been implicated in the biology of various human physiological and pathol......
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Simultaneous determination of long acting LHRH antagonists and its application to high-throughput ph
Aim: Long acting luteinizing hormone-releasing hormone (LHRH) antagonists designed to be protease-resistant were a serie......
目的 探讨血管紧张素受体AT1相关的受体蛋白(APJ)拮抗剂Apelin13(F13A)对肿瘤相关巨噬细胞极化及其诱导的乳腺癌细胞系MCF-7细胞迁......
Aim: To discriminate 32 phenethyl-amines between antagonists and agonists,and predict the activities of these compounds.......
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Bisphenol A exposure alters release of immune and developmental modulators and expression of estroge
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目的 观察螺内酯对肾小球硬化大鼠生长因子-β1(TGF-β1)和结缔组织生长因子(CTGF)表达的影响.方法 40只雄性SD大鼠适应性饲养1周......
目的 观察不同剂量的新斯的明拮抗国产顺式阿曲库铵肌肉松弛的效应.方法 将36例ASA Ⅰ～Ⅱ级择期手术患者分为三组,每组12例,分别给......
Pharmacophore-guided design, synthesis and evaluation of quinazoline-arylpiperazines as new α1-adren
A series of arylpiperazinesquinazoline-2,4-diamine compounds were designed and synthesized based on pharmacophore for ur......
High levels of the neurotoxic beta-amyloid protein (A<em>β</em>) in patients with Alzheimer’s disease present a signif......
AIM: To evaluate the association between acid suppressive drug use and the development of gastric cancer. METHODS: A sys......
目的探讨半胱氨酸白三烯1受体拮抗剂孟鲁司特对慢性支气管炎大鼠气道粘蛋白高分泌的作用.方法气管内注入0.2 mg脂多糖复制模型,采......
目的:通过观察肌电图(EMG)的变化,了解运动员与普通中学生在纵跳过程中,膝关节屈伸肌群工作特点,为运动员科学选材提供依据.方法:3......
从油菜抗、感菌核病品种根际分离具促生和拮抗作用的根际细菌,结果表明从抗病品种中能分离到更多的拮抗和促生菌。其中菌-tu-100 ......
【目的】研究桃树再植病与根际微生物的关系。【方法】以Mфller氰化钾培养基为选择培养基进行桃根际微生物的筛选,采用16SrDNA序......
目的：观察不同剂量的新斯的明拮抗国产阿曲库铵肌松效应。方法：30例ASAⅠ～Ⅱ级择期手术患者分为3组，每组10例，分别给新斯的明20μg／kg(N2......
糖蛋白GP Ⅲb/Ⅲa在血小板表面上的功能表达是血小板抑制剂的最终作用部位。GP Ⅱb/Ⅲa可以与纤维蛋白原桥联而导致血小板凝集。拮......
对自广东、福建、云南、黑龙江、江苏和上海6个省市材料中筛选到的14个细菌菌株与小麦赤霉病菌(F.graminearum)的拮抗作用进行了初......
目的探讨P2X受体拮抗剂（TNP—ATP、PPADS）在大鼠脑缺血性损伤后对神经元的保护作用。方法实验动物随机分为4组：假性手术组、脑梗死组（......
A series of 1,3-substituted 8-styrylxanthines (11a-d) was synthesized, under chemo- and regioselective conditions, in a ......
C5a受体是人和动物体内补体系统的重要组成部分，与C5a结合后介导了众多生物学效应，参与了许多疾病的发生、发展，并在多种病变中起重要......
目的:观察不同浓度的胆汁对胆囊平滑肌运动的影响并初步探讨其作用机理.方法:将肌条置于离体平滑肌灌流肌槽内,用生理记录仪记录肌......
目的研究β-胡萝卜素的抗辐射作用.方法采用30、60、90mg/kgβ-胡萝卜素的剂量对昆明种小鼠进行30 d灌胃,然后用4和8 Gy的60Co-γ......
Laboratory and green house experiments were carried out to evaluate the efficacy of fungicides, biological agents and ho......
Laboratory and green house experiments were carried out to evaluate the efficacy of fungicides, biological agents and ho......
Background: We wanted to determine (via an immunopharmacological approach) whether the c-Jun NH2 terminal kinase (JNK) c......
This review highlights recent advances in pathophysiology and treatment for uremic pruritus, especially focusing on vari......
从山东滕州，临沂等县（市）的烟草，番茄和辣椒根际采集土壤样本１５份，经内分离纯化获得细菌１０２株，放线菌５５株。以烟草赤星病菌，野火病菌和青枯病菌等......
细胞外嘌呤(腺苷、ADP、ATP)及嘧啶(UDP、UTP)为重要的信使分子,通过细胞表面P2受体介导产生不同的生物效应.P2嘌呤受体的概念于19......
观察不同浓度芜花对胆囊平滑肌运动的影响。方法：用８个灌流肌槽同记记录实验动物胆囊肌条的自发收缩活动。结果：（１）芜花水煎剂可增高离体......
This paper analyzes Shakespeare’s different treatment of the male and female antagonists Edmond and Goneril in King Lea......
目的研究褪黑素(MT)对苯妥英(Phe)诱发的胚胎脑组织氧化性损伤有无保护作用.方法妊娠Wistar母鼠于妊娠(GD11～14)ig 0和100 mg·......
促黄体生成激素释放激素（ＬＨＲＨ）活动剂药物已商品化，用于治疗性激素依赖的癌症，ＬＨＲＨ拮抗剂的研究还处于试验阶段。近几年，在寻找高活性，低组胺释放......
Acute ST-Segment Elevation Myocardial Infarction: Combined Intracoronary Low Dose Eptifibatide and T
Aim of the work: To evaluate the efficacy and safety of bolus only intra coronary platelet glyco-protein GP IIb/IIIa rec......
The present review analyses the mechanisms relating heart failure and hyponatremia,describes the association of hyponatr......
Bleeding is the most important complication of oral anticoagulation (OAC) with vitamin K-antagonists. Whilst bleeding is......
<正>近年来,人们利用重组技术从天然生物体内合成了一些新的抗凝药物。这些药物可以弥补华法林功能上的局限性,却有着与华法林相同......
Endothelin receptor antagonists for the treatment of diabetic nephropathy:A meta-analysis and system
BACKGROUND Diabetic nephropathy(DN)is the main cause of chronic kidney disease and endstage renal disease worldwide.Alth......
Phenothiazine vs 5HT3 Antagonist Prophylactic Regimens to Prevent Post‐Anesthesia Care Unit Rescue A
Purpose: Our practitioners are asked to consider a patient’s postoperative nausea and vomiting (PONV) risk profile when......
Growth Hormone Releasing Hormone Receptors Antagonists and Cancers: Do GHRH-R Antagonists Play a Rol
Growth hormone-releasing hormone (GHRH) and its receptors have been implicated in the progression of various tumors such......
Resistant hypertension (RH) has a prevalence of around 12% and is associated with an increased risk of cardiovascular di......
