Molecular Modeling Studies of A3 Adenosine Receptor Modulators Using Machine Learning and Docking Me

来源 :中国上海第七届国际新药发明科技年会 | 被引量 : 0次 | 上传用户:falconcarmack
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  Adenosine receptors (ARs) belong to the G-protein-coupled receptor (GPCR) superfamily and consist of four subtypes referred to as A1,A2A,A2B,and A3.Adenosine receptors have very high sequence similarities among themselves and regulate various biological processes.Therefore,it is important to develop potent and selective modulators of ARs for therapeutic applications.
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